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- A1115 Peptide YY(3-36), PYY, humanTarget: NPY ReceptorsSummary: Y2R激动剂
- A3214 AZD11521 CitationTarget: Aurora KinasesSummary: Aurora B激酶抑制剂
- B7155 BIBP 3226 trifluoroacetateTarget: NPY Receptors|NPFF receptorSummary: 混合NPY Y1和NPFF受体拮抗剂
- A2570 Leupeptin, Microbial中文名: 亮抑酶肽Target: Cathepsins|Calpains|TrypsinsSummary: 丝氨酸和半胱氨酸蛋白酶抑制剂
- A4424 SID 26681509Target: CathepsinsSummary: 人组织蛋白酶L抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A2576 E-642 CitationTarget: Cathepsins|Calpains|PapainsSummary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- N1825 Osthole中文名: 蛇床子素Target: Histamine H1 ReceptorsSummary: 抗肿瘤试剂
- A4122 PHA-680632Target: Aurora Kinases|PLK|FGFRSummary: Aurora激酶抑制剂