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- A1980 SNS-032 (BMS-387032)2 CitationTarget: Cyclin-Dependent KinasesSummary: CDK抑制剂
- A8641 LEE011中文名: 瑞博西利,瑞博西林Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A8385 BMS265246Target: Cyclin-Dependent KinasesSummary: CDK1/2抑制剂
- A8501 PHA-848125中文名: 嘧西利,米尔西利Target: Cyclin-Dependent KinasesSummary: 有效的ATP竞争性CDK抑制剂
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂
- A3266 BS-181Target: Cyclin-Dependent KinasesSummary: CDK7抑制剂
- A2197 Dacarbazine中文名: 达卡巴嗪Target: DNA AlkylatingSummary: 抗肿瘤(恶性黑色素瘤和肉瘤)
- B1299 1-NM-PP1Target: Cyclin-Dependent Kinases|Bcr-Abl|Src|Ca2 /calmodulin-dependent protein kinases (CaMKs)|c-FynSummary: Pp60c-src抑制剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂