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- B2298 Plinabulin (NPI-2358)中文名: 普那布林Target: Vascular Disrupting Agents (VDA)Summary: 血管破坏剂
- B1174 LGX818中文名: 康奈非尼Target: RafSummary: RAF抑制剂
- B1299 1-NM-PP1Target: Cyclin-Dependent Kinases|Bcr-Abl|Src|Ca2 /calmodulin-dependent protein kinases (CaMKs)|c-FynSummary: Pp60c-src抑制剂
- A8328 LDK378中文名: 色瑞替尼Target: ALKSummary: 强效的ALK抑制剂
- A4113 ZM 447439Target: Aurora Kinases|MEK|Src|LckSummary: Aurora激酶抑制剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂