搜索结果: 'research-area pi3k-akt-signaling pi3k-inhibitors'
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- A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: ATP竞争性的Pan-AKT抑制剂
- A5653 AT7867Target: Akt|PKA|p70 rskSummary: Akt1/2/3和p70S6K/PKA的抑制剂
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A8344 K-252cTarget: PKC|PKASummary: 蛋白激酶抑制剂
- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8403 CP-91149Target: Glycogen PhosphorylasesSummary: 糖原磷酸化酶选择性抑制剂
- A4200 Apogossypolone (ApoG2)2 CitationTarget: Bcl-2|Bcl-xl|Mcl-1Summary: Bcl-2的非肽类小分子抑制剂
- B1080 Marinopyrrole ATarget: Mcl-1Summary: 选择性Mcl-1抑制剂
- B3523 Fasudil中文名: 法舒地尔Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 钙拮抗剂