搜索结果: 'research-area gpcr-g-protein protease-activated-receptors'
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- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- B4898 BikininTarget: GSK-3Summary: GSK3抑制剂和油菜素类固醇激活剂
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A8537 Thioridazine HCl中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 ReceptorsSummary: 钙通道蛋白抑制剂
- B2126 Rifabutin中文名: 利福布丁Target: Cytochrome P450 (CYP450)Summary: 抗结核药物
- A3570 LY2090314Target: GSK-3Summary: 有效的GSK-3抑制剂
- A8202 Abiraterone acetate中文名: 乙酸阿比特龙酯Target: Cytochrome P450 (CYP450)Summary: 细胞色素p450 17a1抑制剂