搜索结果: 'research-area endocrinology-and-hormones'
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- A3612 MK-0974Target: CGRP receptorsSummary: CGRP受体拮抗剂
- B1738 Droxidopa中文名: 屈昔多巴Target: adrenergic receptorSummary: 肾上腺素能受体激动剂
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- B1543 Mubritinib (TAK 165)中文名: 木利替尼Target: ErbBSummary: HER2/ErbB2有效抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂
- A3374 Dronedarone中文名: 决奈达隆Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channelSummary: CYP3A4和2D6抑制剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- A3680 OlcegepantTarget: CGRP receptorsSummary: 降钙素基因相关肽(CGRP)的非肽受体,具有有效性和选择性。
- A3146 AGI-6780Target: IDH2Summary: IDH2/R140Q突变抑制剂