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- A8219 Gefitinib (ZD1839)3 Citation中文名: 吉非替尼Target: EGFRSummary: EGFR抑制剂
- A3014 BGJ3981 CitationTarget: FGFRSummary: FGFR抑制剂
- A3011 CHIR-99021 (CT99021)2 CitationTarget: GSK-3Summary: GSK-3抑制剂
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- B1321 OTSSP167Target: MELKSummary: MELK抑制剂
- B1286 AZD7545Target: PDHKSummary: 有效的PDHK选择性抑制剂
- B7794 BMS 3094032 CitationTarget: Fatty-acid-binding proteins (FABPs)Summary: FABP4抑制剂
- A2168 Dovitinib (TKI-258, CHIR-258)2 Citation中文名: 多韦替尼Target: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A3433 Gefitinib hydrochloride中文名: 盐酸吉非替尼Target: EGFRSummary: EGFR有效的抑制剂
- A3258 BMS-833923Target: SmoothenedSummary: Smoothened抑制剂