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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A1302 GSK1904529ATarget: Insulin and Insulin-like ReceptorsSummary: IGF-1R/IR 选择性抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- B1612 Pancuronium dibromide中文名: 泮库溴铵Target: AChRSummary: AChR拮抗剂
- B1620 Tolterodine tartrate中文名: 酒石酸托特罗定Target: AChRSummary: 竞争性毒蕈碱受体拮抗剂
- A5220 Vecuronium Bromide中文名: 维库溴铵Target: AChRSummary: 非去极化神经肌肉松弛剂
- B3703 LB42708Target: FtaseSummary: FTase (法尼基转移酶) 选择性抑制剂
- A8467 Mepenzolate BromideTarget: AChRSummary: mAChR拮抗剂
- A3406 EVP-6124Target: AChRSummary: nAChRs激动剂
- A4302 Rosiglitazone maleate中文名: 马来酸罗格列酮Target: Insulin and Insulin-like ReceptorsSummary: PPARγ激动剂,有效的胰岛素敏化剂