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- A1307 Letrozole中文名: 来曲唑Target: AromatasesSummary: 非甾体类芳香酶抑制剂。
- A4443 Gliotoxin1 CitationTarget: 20S proteasomal chymotrypsin|Geranylgeranyltransferase I|FarnesyltransferaseSummary: 20S蛋白酶体抑制剂
- B1463 KPT-276Target: nuclear export|CRM1Summary: CRM1抑制剂
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A4124 TAK-901Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARGSummary: Aurora A/B抑制剂
- B1382 Anastrozole中文名: 阿那曲唑Target: AromatasesSummary: 芳香酶抑制剂