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- A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53激活剂,阻断Mdm2-p53相互作用。
- A2678 SU112742 CitationTarget: METSummary: C-Met抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- A8533 Terbinafine中文名: 特比萘芬Target: Squalene epoxidasesSummary: 烯丙胺抗真菌剂
- B1901 Butenafine HCl中文名: 盐酸布替萘芬Target: Squalene epoxidasesSummary: 合成苄胺抗真菌剂
- A8325 Tivantinib (ARQ 197)2 CitationTarget: METSummary: C-Met抑制剂
- B5859 Entrectinib中文名: 恩曲替尼Target: Trk Receptors|ALK|ROS1Summary: ALK激酶抑制剂
- B4882 PF-06463922中文名: 劳拉替尼Target: ALK|ROS1Summary: ALK/ROS1的强效选择性抑制剂
- B2047 Terbinafine HCl中文名: 盐酸特比萘芬Target: Squalene epoxidasesSummary: 有效的非竞争性角鲨烯环氧酶抑制剂