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- A4447 2,3-DCPE hydrochlorideTarget: Apoptosis InducersSummary: Bcl-XL蛋白表达下调剂
- A3762 RG71125 CitationTarget: MDM2Summary: MDM2抑制剂
- A4228 Nutlin-3Target: MDM2Summary: MDM2 拮抗剂
- A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2抑制剂
- B5832 Altiratinib1 CitationTarget: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2Summary: c-MET/TIE-2/VEGFR抑制剂
- B3288 APY29Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α变构调节剂
- B5624 STF 083010Target: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1α核酸内切酶抑制剂
- B1874 4μ8C2 CitationTarget: Inositol-requiring enzyme 1 (IRE1)Summary: IRE1 Rnase抑制剂
- N1315 Parthenolide中文名: 小白菊内酯,欧苷菊Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
- A3712 PF-04217903 methanesulfonateTarget: c-METSummary: c-Met抑制剂