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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- B2160 LY2608204Target: GKSummary: GK激活剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- A2917 Flumazenil中文名: 氟马西尼Target: GABAA ReceptorsSummary: 苯二氮卓拮抗剂
- B4904 ACTB-1003Target: VEGFR|FGFR|Tie-2|RSK|p70 S6KSummary: FGFR1抑制剂
- A8435 Furosemide中文名: 呋塞米Target: Na /K /Cl- Symporters (NKCCs)|GABAA ReceptorsSummary: GABAA受体拮抗剂
- N1592 (+)-Bicuculline中文名: 荷包牡丹碱Target: GABAA Receptors|Calcium-Activated Potassium (KCa) ChannelsSummary: GABAA受体拮抗剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性