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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- A3406 EVP-6124Target: AChRSummary: nAChRs激动剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性
- C3869 BQCATarget: AChRSummary: M1毒蕈碱乙酰胆碱受体(mAChR)的正变构调节剂
- A5220 Vecuronium Bromide中文名: 维库溴铵Target: AChRSummary: 非去极化神经肌肉松弛剂
- A3874 Tiotropium BromideTarget: AChRSummary: MAChR M拮抗剂