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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- B2014 Probenecid1 Citation中文名: 丙磺舒Target: Organic anion transporters (OATs)|TRP ChannelSummary: 生物学活性
- A8533 Terbinafine中文名: 特比萘芬Target: Squalene epoxidasesSummary: 烯丙胺抗真菌剂
- B1901 Butenafine HCl中文名: 盐酸布替萘芬Target: Squalene epoxidasesSummary: 合成苄胺抗真菌剂
- B2047 Terbinafine HCl中文名: 盐酸特比萘芬Target: Squalene epoxidasesSummary: 有效的非竞争性角鲨烯环氧酶抑制剂
- A3646 NB-598 hydrochlorideTarget: Squalene epoxidasesSummary: SE抑制剂