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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- B1198 CisaprideTarget: Voltage-gated Potassium (KV) Channels|5-HT4 ReceptorSummary: 5-HT4受体激动剂
- A8534 Terfenadine中文名: 特非那定Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) ChannelsSummary: 组胺H1受体拮抗剂
- A5588 Oligomycin A1 Citation中文名: 寡霉素ATarget: Synthases/SynthetasesSummary: 线粒体ATP合成酶抑制剂
- B3492 Bedaquiline中文名: 贝达喹啉Target: ATP synthaseSummary: 抗结核药物
- B1472 Mizoribine中文名: 咪唑立宾Target: Synthases/SynthetasesSummary: DNA/RNA合成抑制剂
- A2402 Floxuridine中文名: 氟尿苷Target: Synthases/SynthetasesSummary: 抗肿瘤抗代谢物
- B7070 Triacsin CTarget: Synthases/SynthetasesSummary: 酰基辅酶A合成酶抑制剂