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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- N1842 Taxifolin中文名: 紫杉叶素,黄杉素Target: AdipoR2|Opioid receptors
- A4170 EPZ004777Target: DOT1LSummary: DOT1L抑制剂
- B5612 BAY 60-6583Target: Adenosine A2B ReceptorsSummary: A2B受体的强效激动剂
- B1581 EPZ004777 HClTarget: DOT1LSummary: DOT1L抑制剂
- A4166 EPZ56761 CitationTarget: DOT1LSummary: DOT1L抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂