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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- A8660 Cilengitide1 Citation中文名: 西仑吉肽Target: IntegrinsSummary: 整合素αvβ3和αvβ5的抑制剂
- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- A3899 UK-50991 CitationTarget: Monocarboxylate transporters (MCTs)|mitochondrial pyruvate carrier (MPC)Summary: MCTs和MPC抑制剂
- A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1和MCT2抑制剂
- A3145 Afatinib dimaleate中文名: 马来酸阿法替尼Target: EGFR|HER2Summary: EGFR抑制剂
- A8528 TAK-285Target: EGFR|HER2Summary: HER2/EGFR(HER1)抑制剂