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- N1336 Chrysin中文名: 柯因,5,7-二羟黄酮Target: Estrogen and Related Receptors|Hypoxia Inducible Factors (HIFs)Summary: 抗炎和抗肿瘤试剂
- A4347 Methotrexate2 Citation中文名: 甲氨蝶呤Target: Folate AnalogueSummary: 叶酸拮抗剂,抑制DFHR。
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂
- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- B6004 PX-478 2HClTarget: Hypoxia Inducible Factors (HIFs)Summary: HIF-1α抑制剂
- A4383 Tolcapone中文名: 托卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A4168 Entacapone中文名: 恩他卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- B1115 BAY 87-2243Target: Hypoxia Inducible Factors (HIFs)Summary: 有效的HIF-1选择性抑制剂
- B5551 Poly(I:C)Target: Toll-like receptors (TLRs)Summary: Toll样受体3(TLR3)激动剂
- A3444 GS-9620中文名: 维沙莫德Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂