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- A8322 Neratinib (HKI-272)1 Citation中文名: 来那替尼Target: EGFRSummary: HER2/EGFR抑制剂
- A8555 Vandetanib (ZD6474)中文名: 凡德他尼Target: VEGFR|EGFRSummary: VEGFR2/EGFR拮抗剂
- A8357 AG-1478中文名: 酪氨酸磷酸化抑制剂 AG-1478Target: EGFRSummary: EGFR抑制剂
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: 有效的EGFR抑制剂
- B7113 PSB 06126Target: NTPDasesSummary: NTPDase 3抑制剂
- B1079 BMS-303141Target: ATP Citrate LyasesSummary: 有效的ATP-柠檬酸裂合酶抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3194 AST 4871 CitationTarget: RETSummary: RET激酶抑制剂
- A3320 CO-1686 (AVL-301)1 CitationTarget: EGFRSummary: EGFR抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂