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- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- A3358 DeltarasinTarget: Phosphodiesterases (PDEs)Summary: KRAS-PDEδ相互作用抑制剂
- A3021 GDC-0449 (Vismodegib)1 Citation中文名: 维莫德吉Target: P-glycoprotein (P-gp)|HedgehogSummary: Hedgehog拮抗剂
- A3692 OTX-0153 Citation中文名: 比拉瑞塞Target: BromodomainsSummary: BRD抑制剂
- B1564 Ranitidine中文名: 盐酸雷尼替丁Target: Histamine H2 ReceptorsSummary: 组胺H2受体拮抗剂
- B5978 BDA-366Target: Bcl-2Summary: BCL2 BH4 结构域的选择性拮抗剂
- A3023 P0050911 CitationTarget: Ubiquitin-specific proteasesSummary: 泛素特异性蛋白酶7(USP7)抑制剂
- B6026 VR23Target: ProteasomeSummary: 蛋白酶抑制剂
- A3258 BMS-833923Target: SmoothenedSummary: Smoothened抑制剂
- A5424 Fludarabine中文名: 氟达拉滨Summary: DNA合成抑制剂