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- A5057 MGCD-265Target: VEGFR|c-METSummary: Met/Flt/Flk/Ron/Tie-2抑制剂
- A8245 Sorafenib Tosylate1 Citation中文名: 甲苯磺酸索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂
- A1748 Ramelteon1 Citation中文名: 雷美替胺Target: Melatonin ReceptorsSummary: MT1/MT2激动剂
- A3870 TG 100801Target: VEGFR|FGFR|Src|Fyn kinaseSummary: 多激酶抑制剂
- B6274 N-AcetyltryptamineTarget: Melatonin ReceptorsSummary: 褪黑激素受体调节剂
- A8313 RAF265Target: Raf|VEGFRSummary: 多细胞激酶抑制剂
- A8253 PD 173074Target: VEGFR|FGFRSummary: FGFR抑制剂
- A4130 ENMD-2076Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-FmsSummary: Aurora A/Flt3的选择性抑制剂
- A3969 Vatalanib1 Citation中文名: 瓦他拉尼碱Target: VEGFRSummary: 细胞渗透性VEGFR-1/-2抑制剂
- A3009 Sorafenib2 Citation中文名: 索拉非尼Target: Raf|VEGFRSummary: Raf激酶和酪氨酸激酶抑制剂