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- A1805 Imatinib Mesylate (STI571)中文名: 甲磺酸伊马替尼Target: PDGFR|c-Kit|Bcr-AblSummary: Abl/c-kit/PDGFR抑制剂
- A4127 GSK1070916Target: Aurora KinasesSummary: Aurora B/C抑制剂
- A3662 NNC 55-0396Target: Voltage-gated Calcium Channels (CaV)Summary: T型钙离子通道阻断剂
- A8341 Go 6976Target: PKCSummary: PKC α/PKC β1抑制剂
- N1504 Homoharringtonine中文名: 高三尖杉酯碱Target: STATSummary: 细胞毒性生物碱
- A1670 Enzastaurin (LY317615)2 Citation中文名: 恩扎妥林Target: PKCSummary: PKCβ抑制剂
- A3570 LY2090314Target: GSK-3Summary: 有效的GSK-3抑制剂
- B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP抑制剂
- A8217 ICG 0011 CitationSummary: Wnt/β-catenin信号通路的抑制剂
- A1933 Carfilzomib (PR-171)10 Citation中文名: 卡非佐米Target: ProteasomeSummary: 蛋白酶体抑制剂