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- A4374 PF-38451 CitationTarget: FAAHSummary: FAAH抑制剂
- A5112 XL147Target: PI3KSummary: PI3K选择性、可逆的抑制剂
- A8620 AZD-34633 CitationTarget: ALK|Insulin-like growth factors (IGFs)Summary: ALK/IGF1R抑制剂
- A8169 Everolimus (RAD001)8 Citation中文名: 依维莫司Target: mTORSummary: MTOR抑制剂
- A8215 PP 1Target: Src|EGFR|JAK|ZAP-70Summary: Src家族酪氨酸激酶抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂