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- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- A8487 Nocodazole1 Citation中文名: 诺考达唑Target: Microtubules/TubulinsSummary: 微管蛋白产生抑制剂,抗肿瘤剂
- A3433 Gefitinib hydrochloride中文名: 盐酸吉非替尼Target: EGFRSummary: EGFR有效的抑制剂
- B1135 GDC-0623Target: MEKSummary: MEK1抑制剂
- A8169 Everolimus (RAD001)8 Citation中文名: 依维莫司Target: mTORSummary: MTOR抑制剂
- A8340 Cyclopamine1 Citation中文名: 环巴胺Target: SmoothenedSummary: Hedgehog (Hh)信号抑制剂
- A4098 PCI-24781 (CRA-024781)Target: Histone Deacetylases (HDACs)Summary: Pan-HDAC抑制剂
- A8217 ICG 0011 CitationSummary: Wnt/β-catenin信号通路的抑制剂
- A8464 LY21097614 CitationSummary: TβRI/II激酶抑制剂