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- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- B5410 AZ 10606120 dihydrochlorideTarget: P2X ReceptorsSummary: P2X7受体拮抗剂
- B5859 Entrectinib中文名: 恩曲替尼Target: Trk Receptors|ALK|ROS1Summary: ALK激酶抑制剂
- B2189 YM201636Target: PIKfyveSummary: PIKfyve抑制剂
- B2297 GW4417561 CitationTarget: Trk ReceptorsSummary: TrkA抑制剂
- A8303 GNF-5837Target: Trk ReceptorsSummary: Pan-Trk抑制剂