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Signaling Pathways - Octamer-binding transcription factor 4 (Oct4) - Voltage-gated Potassium (KV) Channels - Monocarboxylate transporters (MCTs) - Farnesoid X receptors (FXRs)

10 件产品

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  1. Obeticholic Acid
    B4888 Obeticholic Acid
     2 Citation
    中文名: 奥贝胆酸
    Target: Farnesoid X receptors (FXRs)
    Summary: FXR激动剂
      ≥21.5 mg/mL
      insoluble in H2O
  2. Psora 4
    B7659 Psora 4
     1 Citation
    Target: Voltage-gated Potassium (KV) Channels
    Summary: Kv1.3阻断剂
      ≥15.75 mg/mL
      insoluble in H2O
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. OAC1
    B1994 OAC1
    Target: Octamer-binding transcription factor 4 (Oct4)
    Summary: Oct4激活剂
      ≥9.9 mg/mL
      insoluble in H2O
  5. XL335
    B1528 XL335
    Target: Farnesoid X receptors (FXRs)
    Summary: FXR激动剂
      ≥20.4 mg/mL
      insoluble in H2O
  6. Cisapride
    B1198 Cisapride
    Target: Voltage-gated Potassium (KV) Channels|5-HT4 Receptor
    Summary: 5-HT4受体激动剂
      ≥23.3 mg/mL
      insoluble in H2O
  7. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  8. Lithocholic Acid
    A8463 Lithocholic Acid
    中文名: 石胆酸
    Target: Farnesoid X receptors (FXRs)|Vitamin D receptors (VDRs)|Pregnane X receptor(PXR)
    Summary: 维生素D受体PXR和FXR的激活剂
      ≥12.95 mg/mL
      insoluble in H2O
  9. UK-5099
    A3899 UK-5099
     1 Citation
    Target: Monocarboxylate transporters (MCTs)|mitochondrial pyruvate carrier (MPC)
    Summary: MCTs和MPC抑制剂
      ≥28.8 mg/mL
      insoluble in H2O
  10. AR-C155858
    A3185 AR-C155858
    Target: Monocarboxylate transporters (MCTs)
    Summary: MCT1和MCT2抑制剂
      ≥52.5 mg/mL
      insoluble in H2O

10 件产品

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