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Signaling Pathways - 5-HT receptor - Ubiquitin-activating Enzyme E1 - Voltage-gated Sodium (NaV) Channels

14件产品中的 1-10

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  1. ProTx II
    B5515 ProTx II
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.7通道阻断剂
      Soluble to 1 mg/mL
  2. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  3. Amiloride HCl dihydrate
    B2268 Amiloride HCl dihydrate
    中文名: 盐酸阿米洛利二水合物
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Urokinases
    Summary: 有效上皮钠通道(ENaC)阻断剂
      ≥14.05 mg/mL
      insoluble in H2O
  4. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O
  5. Bupivacaine HCl
    B1420 Bupivacaine HCl
    中文名: 盐酸布比卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 麻醉药
      ≥10.25 mg/mL
      ≥16.23 mg/mL
  6. Phenytoin sodium
    B2272 Phenytoin sodium
    中文名: 苯妥英钠
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 钠通道稳定剂
      ≥11.55 mg/mL
      insoluble in H2O
  7. Proparacaine HCl
    B2274 Proparacaine HCl
    中文名: 盐酸丙美卡因
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: 电压门控钠通道拮抗剂
      ≥14.9 mg/mL
      ≥17.73 mg/mL
  8. MLN4924
    B1036 MLN4924
     5 Citation
    Target: NAE|Ubiquitin-activating Enzyme E1|SUMOylation
    Summary: NAE抑制剂
      ≥22.18 mg/mL
      insoluble in H2O
  9. PYZD-4409
    B1244 PYZD-4409
    Target: Ubiquitin-activating Enzyme E1
    Summary: 泛素激活酶E1抑制剂
      Soluble in DMSO
  10. A-803467
    B2277 A-803467
    Target: Voltage-gated Sodium (NaV) Channels
    Summary: NaV1.8通道阻断剂
      ≥13.95 mg/mL
      insoluble in H2O

14件产品中的 1-10

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