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Signaling Pathways - L3MBTL - PKG - Voltage-gated Potassium (KV) Channels - CCR

10 件产品

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  1. Psora 4
    B7659 Psora 4
     1 Citation
    Target: Voltage-gated Potassium (KV) Channels
    Summary: Kv1.3阻断剂
      ≥15.75 mg/mL
      insoluble in H2O
  2. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  3. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  4. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  5. Cisapride
    B1198 Cisapride
    Target: Voltage-gated Potassium (KV) Channels|5-HT4 Receptor
    Summary: 5-HT4受体激动剂
      ≥23.3 mg/mL
      insoluble in H2O
  6. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  7. Maraviroc
    A8311 Maraviroc
     2 Citation
    中文名: 马拉维若
    Target: CCR
    Summary: CCR5选择性拮抗剂,抗逆转录病毒药物
      ≥25.7 mg/mL
      insoluble in H2O
  8. GSK690693
    A5072 GSK690693
    Target: Akt|PKC|PKG|PKA|Prk
    Summary: ATP竞争性的Pan-AKT抑制剂
      ≥21.25 mg/mL
      insoluble in H2O
  9. UNC1215
    A3901 UNC1215
     1 Citation
    Target: L3MBTL
    Summary: 甲基赖氨酸的化学探针
      ≥26.05 mg/mL
      insoluble in H2O
  10. INCB3344
    A3494 INCB3344
    Target: CCR
    Summary: CCR2趋化因子受体拮抗剂
      ≥25.9 mg/mL
      insoluble in H2O

10 件产品

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