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Signaling Pathways - KDM - CETP - adrenergic receptor - P2X Receptors

11件产品中的 1-10

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  1. TC-E 5002
    B4930 TC-E 5002
    Target: KDM
    Summary: 选择性组蛋白去甲基化酶KDM2/7亚家族抑制剂
      Soluble in DMSO
  2. AZ 10606120 dihydrochloride
    B5410 AZ 10606120 dihydrochloride
    Target: P2X Receptors
    Summary: P2X7受体拮抗剂
      <49.55 mg/mL
      <12.39 mg/mL
  3. Epinephrine Bitartrate
    B1358 Epinephrine Bitartrate
    中文名: 酒石酸肾上腺素
    Target: adrenergic receptor
    Summary: 肾上腺素能受体激动剂
      ≥16.66 mg/mL
      ≥22.9 mg/mL
  4. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O
  5. Quetiapine
    A3744 Quetiapine
    中文名: 喹硫平
    Target: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptor
    Summary: 多巴胺受体拮抗剂
      ≥19.18 mg/mL
      insoluble in H2O
  6. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  7. Daminozide
    A3348 Daminozide
    中文名: 丁酰肼
    Target: KDM|PHF
    Summary: KDM2A抑制剂
      ≥7.3 mg/mL
      ≥21.4 mg/mL
  8. A-740003
    A3136 A-740003
    Target: P2X Receptors
    Summary: P2X7受体拮抗剂
      ≥23.73 mg/mL
      insoluble in H2O
  9. Evacetrapib (LY2484595)
    A4377 Evacetrapib (LY2484595)
    Target: CETP
    Summary: 强效的CETP选择性抑制剂
      ≥32.1 mg/mL
      insoluble in H2O
  10. Anacetrapib (MK-0859)
    A4375 Anacetrapib (MK-0859)
     1 Citation
    中文名: 安塞曲匹
    Target: CETP
    Summary: RhCETP/突变型 CETP(C13S) 抑制剂
      ≥31.9 mg/mL
      insoluble in H2O

11件产品中的 1-10

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