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Signaling Pathways - endothelin receptor - Factor Xa - NOS - sodium channel

11件产品中的 1-10

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  1. FR 139317
    B5082 FR 139317
    Target: endothelin receptor
    Summary: 选择性ETA内皮素受体拮抗剂
      Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
  2. L-NIO dihydrochloride
    B6345 L-NIO dihydrochloride
    Target: NOS
    Summary: 一氧化氮(NO)合酶抑制剂
      <24.61 mg/mL
  3. Diphenyleneiodonium chloride
    B6326 Diphenyleneiodonium chloride
    中文名: 二苯基氯化碘盐
    Target: NADPH Oxidases|NOS|GPR3
    Summary: iNOS和eNOS抑制剂,GPR3激动剂
      ≥6.99 mg/mL
      insoluble in H2O
  4. 7-Nitroindazole
    B6369 7-Nitroindazole
    中文名: 硝基吲唑
    Target: NOS
    Summary: nNOS抑制剂
      ≥5.85 mg/mL
      insoluble in H2O
  5. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  6. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  7. Otamixaban
    A3690 Otamixaban
    中文名: 奥米沙班
    Target: Factor Xa
    Summary: 因子Xa抑制剂
      ≥22.35 mg/mL
      insoluble in H2O
  8. Edoxaban
    A3381 Edoxaban
    中文名: 依度沙班
    Target: Factor Xa
    Summary: 因子Xa抑制剂
      ≥27.3 mg/mL
      insoluble in H2O
  9. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  10. 5-R-Rivaroxaban
    A3126 5-R-Rivaroxaban
    中文名: 5-R-利伐沙班
    Target: Factor Xa
    Summary: 因子Xa(FXa)抑制剂
      ≥20.85 mg/mL
      insoluble in H2O

11件产品中的 1-10

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