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Signaling Pathways - endothelin receptor - Hck - c-MET - Calcium-Activated Potassium (KCa) Channels

14件产品中的 1-10

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  1. Altiratinib
    B5832 Altiratinib
     1 Citation
    Target: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2
    Summary: c-MET/TIE-2/VEGFR抑制剂
      ≥21.55 mg/mL
      insoluble in H2O
  2. FR 139317
    B5082 FR 139317
    Target: endothelin receptor
    Summary: 选择性ETA内皮素受体拮抗剂
      Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
  3. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  4. PP121
    B2172 PP121
    Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|Hck
    Summary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
      ≥15.95 mg/mL
      insoluble in H2O
  5. INCB28060
    A8448 INCB28060
    中文名: 苯扎米特
    Target: c-MET
    Summary: C-Met抑制剂
      ≥5.15 mg/mL
      insoluble in H2O
  6. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  7. MGCD-265
    A5057 MGCD-265
    Target: VEGFR|c-MET
    Summary: Met/Flt/Flk/Ron/Tie-2抑制剂
      ≥25.9 mg/mL
      insoluble in H2O
  8. CP-724714
    A2412 CP-724714
    Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1R
    Summary: 有效的HER2选择性抑制剂
      ≥23.5 mg/mL
      insoluble in H2O
  9. PF-04217903
    A5096 PF-04217903
    Target: c-MET
    Summary: C-Met的选择性和ATP竞争性抑制剂
      ≥18.6 mg/mL
      insoluble in H2O
  10. PHA-665752
    A2307 PHA-665752
     1 Citation
    Target: c-MET
    Summary: c-Met的ATP竞争性、有效的、选择性抑制剂
      ≥32.1 mg/mL
      insoluble in H2O

14件产品中的 1-10

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