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Signaling Pathways - c-RET - p53 - Urokinases - potassium channel

14件产品中的 1-10

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  1. G-749
    A8889 G-749
    Target: Aurora Kinases|FLT3|c-RET
    Summary: FLT3抑制剂
      ≥26.05 mg/mL
      insoluble in H2O
  2. Amiloride HCl dihydrate
    B2268 Amiloride HCl dihydrate
    中文名: 盐酸阿米洛利二水合物
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Urokinases
    Summary: 有效上皮钠通道(ENaC)阻断剂
      ≥14.05 mg/mL
      insoluble in H2O
  3. Pifithrin-μ
    A4482 Pifithrin-μ
     1 Citation
    Target: Autophagy|p53|HSP70
    Summary: p53结合抑制剂,抗凋亡。
      ≥18.1 mg/mL
      insoluble in H2O
  4. PRIMA-1
    A4483 PRIMA-1
    Target: p53
    Summary: BAX抑制剂
      ≥9.1 mg/mL
      ≥110.6 mg/mL
  5. PhiKan 083
    A4481 PhiKan 083
    Target: p53
    Summary: P53稳定剂
      <27.48 mg/mL
      <13.74 mg/mL
  6. 4-Chlorophenylguanidine hydrochloride
    A4445 4-Chlorophenylguanidine hydrochloride
    Target: Urokinases
    Summary: 尿激酶(urokinase)抑制剂
      Soluble to 100 mM in H2O
  7. Regorafenib hydrochloride
    A3750 Regorafenib hydrochloride
    中文名: 瑞戈非尼盐酸盐
    Target: Raf|VEGFR|PDGFR|c-Kit|c-RET
    Summary: 酪氨酸激酶抑制剂
      ≥25.95 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Tenovin-1
    A4203 Tenovin-1
    Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21
    Summary: SIRT2 抑制剂,p53激活剂
      ≥15 mg/mL
      insoluble in H2O
  10. JNJ-26854165 (Serdemetan)
    A4204 JNJ-26854165 (Serdemetan)
     1 Citation
    Target: p53|HDM2 ubiquitin ligase
    Summary: P53激活剂,阻断Mdm2-p53相互作用。
      ≥14.8 mg/mL
      insoluble in H2O

14件产品中的 1-10

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