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Signaling Pathways - NAE - Lyn - sodium channel - Nrf2

10 件产品

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  1. SU6656
    B5839 SU6656
    Target: Src|Lyn|YES|Fyn
    Summary: Src 酪氨酸激酶抑制剂
      ≥18.55 mg/mL
      insoluble in H2O
  2. Omaveloxolone (RTA-408)
    B3576 Omaveloxolone (RTA-408)
    Target: Nrf2
    Summary: Nrf2激活剂
      ≥55.5 mg/mL
      insoluble in H2O
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  5. MLN4924
    B1036 MLN4924
     5 Citation
    Target: NAE|Ubiquitin-activating Enzyme E1|SUMOylation
    Summary: NAE抑制剂
      ≥22.18 mg/mL
      insoluble in H2O
  6. Masitinib (AB1010)
    A2942 Masitinib (AB1010)
    中文名: 马赛替尼
    Target: PDGFR|c-Kit|Lyn
    Summary: 酪氨酸激酶抑制剂
      ≥24.95 mg/mL
      insoluble in H2O
  7. MLN4924 HCl salt
    A3629 MLN4924 HCl salt
    Target: NAE
    Summary: NAE inhibitor
      Soluble in DMSO
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Curcumin
    A3335 Curcumin
     1 Citation
    中文名: 姜黄素
    Target: Histone Deacetylases (HDACs)|Nrf2|Histone Acetyltransferases (HATs)|Tyrosinases
    Summary: Tyrosinase(酪氨酸酶)抑制剂
      ≥36.8 mg/mL
      insoluble in H2O
  10. Bardoxolone methyl
    A3221 Bardoxolone methyl
    中文名: 甲基巴多索隆
    Target: Nrf2
    Summary: IKK抑制剂,强效的抗氧化炎性反应调节剂。
      ≥25.3 mg/mL
      insoluble in H2O

10 件产品

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