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Signaling Pathways - 5-HT4 Receptors - Papains - Melanocortin (MC) Receptors - P-glycoprotein (P-gp)

10 件产品

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  1. Papain Inhibitor
    A1035 Papain Inhibitor
    Target: Papains
    Summary: 木瓜蛋白酶抑制剂
      ≥45.1 mg/mL
      ≥90.4 mg/mL
  2. LY335979 (Zosuquidar 3HCL)
    A8549 LY335979 (Zosuquidar 3HCL)
     1 Citation
    中文名: 唑喹达三盐酸盐
    Target: P-glycoprotein (P-gp)
    Summary: Pgb(P糖蛋白)抑制剂
      ≥17.1 mg/mL
      ≥31.9 mg/mL
  3. Mosapride Citrate
    A1334 Mosapride Citrate
    中文名: 莫沙必利柠檬酸盐
    Target: 5-HT3 Receptors|5-HT4 Receptors
    Summary: 5-HT受体激动剂
      ≥30.7 mg/mL
      insoluble in H2O
  4. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  5. Tariquidar methanesulfonate, hydrate
    A3859 Tariquidar methanesulfonate, hydrate
    中文名: 他立喹达二甲磺酸盐六水合物
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥56.2 mg/mL
      insoluble in H2O
  6. Elacridar
    A3384 Elacridar
    中文名: 依克立达
    Target: P-glycoprotein (P-gp)
    Summary: BCRP抑制剂
      ≥56.4 mg/mL
      insoluble in H2O
  7. Agouti-related Protein (AGRP) (25-82), human
    A1134 Agouti-related Protein (AGRP) (25-82), human
    Target: Melanocortin (MC) Receptors
    Summary: 刺鼠相关肽(25-82)
      insoluble in DMSO
      ≥100 mg/mL
  8. Tariquidar
    A8208 Tariquidar
     2 Citation
    中文名: 他立喹达
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥16.17 mg/mL
      insoluble in H2O
  9. E-64
    A2576 E-64
     2 Citation
    Target: Cathepsins|Calpains|Papains
    Summary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
      ≥53.6 mg/mL
      ≥49.1 mg/mL
  10. GDC-0449 (Vismodegib)
    A3021 GDC-0449 (Vismodegib)
     1 Citation
    中文名: 维莫德吉
    Target: P-glycoprotein (P-gp)|Hedgehog
    Summary: Hedgehog拮抗剂
      ≥21.08 mg/mL
      insoluble in H2O

10 件产品

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