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Signaling Pathways - Calcium-Activated Potassium (KCa) Channels - 5-HT2 Receptor - SUMOylation - MK2

10 件产品

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  1. MK2 Inhibitor IV
    C5545 MK2 Inhibitor IV
    Target: MK2
    Summary: 高选择性、非ATP竞争性MK2抑制剂
      insoluble in DMSO
      ≥37.4 mg/mL
  2. CMPD-1
    B6962 CMPD-1
    Target: Microtubules/Tubulins|MK2
    Summary: p38α介导的MK2a磷酸化的抑制剂
      <34.94 mg/mL
      <34.94 mg/mL
  3. SCH 23390 hydrochloride
    B6506 SCH 23390 hydrochloride
    Target: dopamine receptor|5-HT1 Receptor|5-HT2 Receptor
    Summary: 多巴胺受体拮抗剂
      Soluble to 100 mM in sterile water and to 50 mM in ethanol
  4. Methylergometrine maleate
    B6347 Methylergometrine maleate
    中文名: 马来酸甲麦角新碱
    Target: 5-HT1 Receptor|5-HT2 Receptor
    Summary: 5-HT1/5-HT2受体拮抗剂
      Soluble to 25 mM in H2O
  5. PF-3644022
    B5549 PF-3644022
    Target: MK2
    Summary: MK2抑制剂
      <14.98 mg/mL
  6. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  7. MLN4924
    B1036 MLN4924
     5 Citation
    Target: NAE|Ubiquitin-activating Enzyme E1|SUMOylation
    Summary: NAE抑制剂
      ≥22.18 mg/mL
      insoluble in H2O
  8. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  9. TRAM-34
    A1888 TRAM-34
    Target: Calcium-Activated Potassium (KCa) Channels
    Summary: KCa3.1阻断剂
      ≥17.25 mg/mL
      insoluble in H2O
  10. PHA-767491
    A3721 PHA-767491
    Target: Cyclin-Dependent Kinases|MK2|Cdc7
    Summary: Cdc7 / CDK9抑制剂
      ≥10.65 mg/mL
      insoluble in H2O

10 件产品

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