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Signaling Pathways - CK1 - AChE - sodium channel - CB2 Receptors

10 件产品

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  1. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  2. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  3. Donepezil HCl
    B1602 Donepezil HCl
    中文名: 盐酸多奈哌齐
    Target: AChE
    Summary: AChE抑制剂
      insoluble in DMSO
      ≥10.4 mg/mL
  4. BML-190
    B1425 BML-190
    中文名: 吲哚美辛吗啉代酰胺
    Target: CB2 Receptors
    Summary: CB2受体的配体
      ≥42.7 mg/mL
      insoluble in H2O
  5. Rimonabant
    B1429 Rimonabant
     3 Citation
    中文名: 利莫那班
    Target: CB1 Receptors|CB2 Receptors
    Summary: CB1 受体拮抗剂
      ≥23.19 mg/mL
      insoluble in H2O
  6. PF-670462
    A3719 PF-670462
    Target: CK1
    Summary: CK1 ε/δ抑制剂
      ≥20.5 mg/mL
      ≥94 mg/mL
  7. Galanthamine
    A3423 Galanthamine
     2 Citation
    中文名: 加兰他敏
    Target: AChE
    Summary: 乙酰胆碱酯酶抑制剂
      ≥14.37 mg/mL
      ≥14.43 mg/mL
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. D4476
    A3342 D4476
     1 Citation
    Target: CK1
    Summary: CK1/ALK5抑制剂
      ≥19.9 mg/mL
      insoluble in H2O
  10. (-)-Huperzine A
    A1932 (-)-Huperzine A
    中文名: 石杉碱甲
    Target: NMDA Receptors|AChE
    Summary: NMDA受体拮抗剂/AChE抑制剂
      ≥12.12 mg/mL
      insoluble in H2O

10 件产品

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