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Signaling Pathways - Pyruvate dehydrogenases (PDH) - Voltage-gated Potassium (KV) Channels - sterol demethylase - TRP Channel

10 件产品

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  1. FG2216
    B5851 FG2216
    Target: Pyruvate dehydrogenases (PDH)
    Summary: HIF-脯氨酰羟化酶抑制剂
      ≥14.05 mg/mL
      insoluble in H2O
  2. Psora 4
    B7659 Psora 4
     1 Citation
    Target: Voltage-gated Potassium (KV) Channels
    Summary: Kv1.3阻断剂
      ≥15.75 mg/mL
      insoluble in H2O
  3. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  4. Cisapride
    B1198 Cisapride
    Target: Voltage-gated Potassium (KV) Channels|5-HT4 Receptor
    Summary: 5-HT4受体激动剂
      ≥23.3 mg/mL
      insoluble in H2O
  5. Icilin
    B1055 Icilin
    Target: TRP Channel
    Summary: TRPM8/ hENaCδ激动剂
      ≥11.05 mg/mL
      insoluble in H2O
  6. Terfenadine
    A8534 Terfenadine
    中文名: 特非那定
    Target: Voltage-gated Potassium (KV) Channels|Histamine H1 Receptors|Inward Rectifier Potassium (Kir) Channels
    Summary: 组胺H1受体拮抗剂
      ≥18 mg/mL
      insoluble in H2O
  7. AMG-517
    A1174 AMG-517
    Target: TRP Channel
    Summary: TRPV1拮抗剂
      ≥21.5 mg/mL
      insoluble in H2O
  8. Posaconazole
    A1718 Posaconazole
    中文名: 泊沙康唑
    Target: Cytochrome P450 (CYP450)|sterol demethylase
    Summary: 甾醇 C14ɑ去甲基化酶抑制剂
      ≥35.04 mg/mL
      insoluble in H2O
  9. Nonivamide (Capsaicin Analog)
    A3278 Nonivamide (Capsaicin Analog)
     1 Citation
    中文名: 香草壬酰胺
    Target: TRP Channel
    Summary: TRPV1受体激动剂
      ≥15.27 mg/mL
      insoluble in H2O
  10. CPI-613
    A4333 CPI-613
     1 Citation
    Target: Pyruvate dehydrogenases (PDH)
    Summary: PDH/α-KGDH抑制剂
      ≥19.45 mg/mL
      insoluble in H2O

10 件产品

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