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Signaling Pathways - EP300 - HIV - calcium uptake - P-glycoprotein (P-gp)

10 件产品

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  1. LY335979 (Zosuquidar 3HCL)
    A8549 LY335979 (Zosuquidar 3HCL)
     1 Citation
    中文名: 唑喹达三盐酸盐
    Target: P-glycoprotein (P-gp)
    Summary: Pgb(P糖蛋白)抑制剂
      ≥17.1 mg/mL
      ≥31.9 mg/mL
  2. Ranolazine
    A8510 Ranolazine
     1 Citation
    中文名: 雷诺嗪
    Target: calcium uptake
    Summary: 抗缺血
      ≥17.4 mg/mL
      insoluble in H2O
  3. SGC-CBP30
    A4491 SGC-CBP30
     2 Citation
    Target: CREBBP|EP300
    Summary: CREBBP/EP300 bromodomain抑制剂
      ≥20.05 mg/mL
      ≥4.67 mg/mL
  4. I-CBP 112
    A4490 I-CBP 112
    Target: CREBBP|EP300
    Summary: CBP/EP300 bromodomain抑制剂
      ≥49.6 mg/mL
      insoluble in H2O
  5. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  6. Tariquidar methanesulfonate, hydrate
    A3859 Tariquidar methanesulfonate, hydrate
    中文名: 他立喹达二甲磺酸盐六水合物
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥56.2 mg/mL
      insoluble in H2O
  7. Elacridar
    A3384 Elacridar
    中文名: 依克立达
    Target: P-glycoprotein (P-gp)
    Summary: BCRP抑制剂
      ≥56.4 mg/mL
      insoluble in H2O
  8. Betulinic acid
    A3237 Betulinic acid
    中文名: 白桦脂酸,桦木酸
    Target: Aminopeptidases|Topoisomerases|HIV
    Summary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
      ≥22.85 mg/mL
      insoluble in H2O
  9. Tariquidar
    A8208 Tariquidar
     2 Citation
    中文名: 他立喹达
    Target: P-glycoprotein (P-gp)
    Summary: P-糖蛋白抑制剂
      ≥16.17 mg/mL
      insoluble in H2O
  10. GDC-0449 (Vismodegib)
    A3021 GDC-0449 (Vismodegib)
     1 Citation
    中文名: 维莫德吉
    Target: P-glycoprotein (P-gp)|Hedgehog
    Summary: Hedgehog拮抗剂
      ≥21.08 mg/mL
      insoluble in H2O

10 件产品

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