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Signaling Pathways - Bcl-2 - Voltage-gated Calcium Channels (CaV) - MK2 - ALK

34件产品中的 1-10

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  1. MK2 Inhibitor IV
    C5545 MK2 Inhibitor IV
    Target: MK2
    Summary: 高选择性、非ATP竞争性MK2抑制剂
      insoluble in DMSO
      ≥37.4 mg/mL
  2. BDA-366
    B5978 BDA-366
    Target: Bcl-2
    Summary: BCL2 BH4 结构域的选择性拮抗剂
      ≥50.4 mg/mL
      insoluble in H2O
  3. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  4. (+)-Apogossypol
    B4902 (+)-Apogossypol
    中文名: 變棉子酚,阿朴棉子酚,变棉子酚
    Target: Bcl-2
    Summary: Bcl-2家族蛋白抑制剂
      ≥16.2 mg/mL
      insoluble in H2O
  5. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  6. CMPD-1
    B6962 CMPD-1
    Target: Microtubules/Tubulins|MK2
    Summary: p38α介导的MK2a磷酸化的抑制剂
      <34.94 mg/mL
      <34.94 mg/mL
  7. PF-3644022
    B5549 PF-3644022
    Target: MK2
    Summary: MK2抑制剂
      <14.98 mg/mL
  8. SNX 482
    B5351 SNX 482
    Target: Voltage-gated Calcium Channels (CaV)
    Summary: 电压依赖性R型CaV2.3钙通道阻滞剂
      Soluble in H2O
  9. Amiloride HCl dihydrate
    B2268 Amiloride HCl dihydrate
    中文名: 盐酸阿米洛利二水合物
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Urokinases
    Summary: 有效上皮钠通道(ENaC)阻断剂
      ≥14.05 mg/mL
      insoluble in H2O
  10. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O

34件产品中的 1-10

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