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Signaling Pathways - NUAK2 - Cytochrome P450 (CYP450) - MK2 - Cell Experiments

12件产品中的 1-10

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  1. MK2 Inhibitor IV
    C5545 MK2 Inhibitor IV
    Target: MK2
    Summary: 高选择性、非ATP竞争性MK2抑制剂
      insoluble in DMSO
      ≥37.4 mg/mL
  2. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  3. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  4. Clotrimazole
    A8401 Clotrimazole
     2 Citation
    中文名: 克霉唑
    Target: Cytochrome P450 (CYP450)
    Summary: 抗真菌化合物
      ≥28.1 mg/mL
      insoluble in H2O
  5. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  6. Posaconazole
    A1718 Posaconazole
    中文名: 泊沙康唑
    Target: Cytochrome P450 (CYP450)|sterol demethylase
    Summary: 甾醇 C14ɑ去甲基化酶抑制剂
      ≥35.04 mg/mL
      insoluble in H2O
  7. PHA-767491
    A3721 PHA-767491
    Target: Cyclin-Dependent Kinases|MK2|Cdc7
    Summary: Cdc7 / CDK9抑制剂
      ≥10.65 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Clarithromycin
    A4322 Clarithromycin
    中文名: 克拉霉素
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A抑制剂
      ≥31.2 mg/mL
      insoluble in H2O
  10. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O

12件产品中的 1-10

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