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- B5851 FG2216Target: Pyruvate dehydrogenases (PDH)Summary: HIF-脯氨酰羟化酶抑制剂
- B1373 Phenformin HCl1 Citation中文名: 盐酸苯乙双胍,盐酸苯乙福明Target: AMPKSummary: 抗糖尿病
- B3252 Dorsomorphin (Compound C)5 CitationTarget: AMPKSummary: AMPK抑制剂
- A4333 CPI-6131 CitationTarget: Pyruvate dehydrogenases (PDH)Summary: PDH/α-KGDH抑制剂
- A4377 Evacetrapib (LY2484595)Target: CETPSummary: 强效的CETP选择性抑制剂
- A4375 Anacetrapib (MK-0859)1 Citation中文名: 安塞曲匹Target: CETPSummary: RhCETP/突变型 CETP(C13S) 抑制剂