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- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- A3291 CCT241533Target: ChkSummary: 有效的Chk2抑制剂
- B1579 JIB-041 CitationTarget: Histone DemethylasesSummary: Jumonji组蛋白去甲基化酶抑制剂
- B1054 Resiquimod (R-848)2 Citation中文名: 雷西莫特,瑞喹莫德Target: Toll-like receptors (TLRs)Summary: 免疫应答调节剂
- B5551 Poly(I:C)Target: Toll-like receptors (TLRs)Summary: Toll样受体3(TLR3)激动剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂