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- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- A2402 Floxuridine中文名: 氟尿苷Target: Synthases/SynthetasesSummary: 抗肿瘤抗代谢物
- A3446 GSK1265 CitationTarget: EZH2Summary: EZH2抑制剂
- A3214 AZD11521 CitationTarget: Aurora KinasesSummary: Aurora B激酶抑制剂
- N1620 Ginsenoside Rb1中文名: 人参皂苷 Rb1Summary: 抗增殖剂
- A1947 MEK162 (ARRY-162, ARRY-438162)中文名: 贝美替尼Target: MEKSummary: MEK1/2抑制剂
- A3859 Tariquidar methanesulfonate, hydrate中文名: 他立喹达二甲磺酸盐六水合物Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A2173 SC 1441 CitationTarget: GlycoproteinsSummary: Gp130抑制剂
- A8225 EzatiostatTarget: Gutathione S-transferaseSummary: (GST) P1-1抑制剂
- A8557 TAE226 (NVP-TAE226)1 CitationTarget: FAKSummary: 强效的ATP竞争性FAK抑制剂