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- A5573 Pimasertib (AS-703026)Target: MEKSummary: MEK1/2抑制剂
- B1621 TAK-733Target: MEKSummary: MEK变构位点抑制剂
- A4386 Elesclomol (STA-4783)3 Citation中文名: 伊利司莫Summary: 氧化应激/细胞凋亡诱导剂
- B3704 Nexturastat ATarget: Histone Deacetylases (HDACs)Summary: HDAC6抑制剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- N1375 Solamargine中文名: 澳洲茄边碱,边缘茄碱Summary: 细胞毒性剂
- A3170 AM9662 CitationTarget: LPA ReceptorsSummary: LPA1拮抗剂