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- A4313 Cobicistat (GS-9350)中文名: 可比司他Target: Cytochrome P450 (CYP450)Summary: CYP3A的选择性抑制剂
- B2094 Fluconazole中文名: 氟康唑Target: Cytochrome P450 (CYP450)Summary: 三唑抗真菌剂
- B6227 Kynurenic acid中文名: 犬尿酸Target: EAA receptorSummary: 广谱EAA拮抗剂
- B7590 Quinidine中文名: 奎尼丁Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)Summary: 降低Na+和K+通道电流
- A8432 Fenticonazole Nitrate中文名: 硝酸芬替康唑Target: Cytochrome P450 (CYP450)|Synthases/SynthetasesSummary: 抗真菌药
- A3327 Costunolide中文名: 木香烃内酯Target: FPTase|TelomerasesSummary: BMM分化抑制剂
- A8401 Clotrimazole2 Citation中文名: 克霉唑Target: Cytochrome P450 (CYP450)Summary: 抗真菌化合物
- A4379 Lonafarnib中文名: 洛那法尼Target: FPTaseSummary: 高效且具有选择性的法尼基转移酶抑制剂
- A1718 Posaconazole中文名: 泊沙康唑Target: Cytochrome P450 (CYP450)|sterol demethylaseSummary: 甾醇 C14ɑ去甲基化酶抑制剂
- A4322 Clarithromycin中文名: 克拉霉素Target: Cytochrome P450 (CYP450)Summary: CYP3A抑制剂