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- A4313 Cobicistat (GS-9350)中文名: 可比司他Target: Cytochrome P450 (CYP450)Summary: CYP3A的选择性抑制剂
- B2094 Fluconazole中文名: 氟康唑Target: Cytochrome P450 (CYP450)Summary: 三唑抗真菌剂
- B7590 Quinidine中文名: 奎尼丁Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)Summary: 降低Na+和K+通道电流
- A8432 Fenticonazole Nitrate中文名: 硝酸芬替康唑Target: Cytochrome P450 (CYP450)|Synthases/SynthetasesSummary: 抗真菌药
- B4899 BLZ9451 CitationTarget: CSF-1RSummary: CSF-1R激酶抑制剂
- A1655 GW25801 CitationTarget: CSF-1RSummary: CFMS激酶/CSF-1R抑制剂
- A3022 Pazopanib (GW-786034)中文名: 帕唑帕尼Target: CSF-1R|VEGFR|PDGFR|c-Kit|FGFRSummary: (GW-786034)VEGFR/PDGFR/FGFR 的抑制剂。
- A8401 Clotrimazole2 Citation中文名: 克霉唑Target: Cytochrome P450 (CYP450)Summary: 抗真菌化合物
- B1500 I-BET151 (GSK1210151A)2 CitationTarget: Bromodomain and Extra-Terminal motif (BET)Summary: BET的选择性抑制剂
- A1718 Posaconazole中文名: 泊沙康唑Target: Cytochrome P450 (CYP450)|sterol demethylaseSummary: 甾醇 C14ɑ去甲基化酶抑制剂