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- A2877 Camptothecin1 Citation中文名: 喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- B2295 Pirarubicin1 Citation中文名: 吡柔比星Target: TopoisomerasesSummary: 拓扑异构酶II抑制剂,蒽环类抗生素
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- B7382 Ellipticine中文名: 玫瑰树碱,椭圆玫瑰树碱Target: TopoisomerasesSummary: DNA拓扑异构酶II抑制剂
- N2133 7-Ethyl-10-hydroxycamptothecinTarget: TopoisomerasesSummary: TOPO I抑制剂
- A4536 Fostriecin sodium saltTarget: PP1|PP2A|Topoisomerases|PP4Summary: 抗肿瘤抗生素
- B1036 MLN49245 CitationTarget: NAE|Ubiquitin-activating Enzyme E1|SUMOylationSummary: NAE抑制剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: ATP竞争性的Pan-AKT抑制剂
- A8344 K-252cTarget: PKC|PKASummary: 蛋白激酶抑制剂