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- A1877 XAV-9391 CitationTarget: TNKSSummary: Tankyrase 1/2抑制剂
- B4892 TAI-1Target: Hec1Summary: Hec1抑制剂
- A3899 UK-50991 CitationTarget: Monocarboxylate transporters (MCTs)|mitochondrial pyruvate carrier (MPC)Summary: MCTs和MPC抑制剂
- A3185 AR-C155858Target: Monocarboxylate transporters (MCTs)Summary: MCT1和MCT2抑制剂