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- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂
- A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90抑制剂
- B5743 SR 2211Target: Retinoic acid-related Orphan Receptors (RORs)Summary: RORγ反向激动剂
- B7393 GeduninTarget: HSP90Summary: 天然的Hsp90抑制剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A4064 NVP-BEP800Target: HSP90Summary: 全合成的HSP90β口服抑制剂
- B2087 Ciclopirox中文名: 环吡酮胺Target: HydroxylasesSummary: 广谱抗真菌剂
- A4061 IPI-504 (Retaspimycin hydrochloride)3 Citation中文名: 瑞他霉素盐酸盐Target: HSP90Summary: Hsp90抑制剂
- A4056 AT13387Target: HSP90Summary: Hsp90抑制剂
- B4920 EC 144Target: HSP90Summary: Hsp90抑制剂