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- A3170 AM9662 CitationTarget: LPA ReceptorsSummary: LPA1拮抗剂
- B1963 Lomustine1 Citation中文名: 洛莫司汀Target: RNA synthesisSummary: 抗肿瘤药
- B3941 Talabostat mesylate2 CitationTarget: DPP-4Summary: DPP4抑制剂
- B2186 GSK2636771Target: PI3KSummary: PIK3抑制剂
- A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90抑制剂
- A4094 MC15683 CitationTarget: Histone Deacetylases (HDACs)Summary: II类HDAC抑制剂
- B4900 Indoximod (NLG-8189)Summary: 吲哚胺2,3-双加氧酶(IDO)途径抑制剂
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- N1375 Solamargine中文名: 澳洲茄边碱,边缘茄碱Summary: 细胞毒性剂
- B1174 LGX818中文名: 康奈非尼Target: RafSummary: RAF抑制剂